Sentence examples for series displaying from inspiring English sources

Compounds 12a, 12d, and 28 are the most active derivatives in this series, displaying activity comparable to that of retapamulin and BC-3781.

He has been a one-man show against the marauding English in this series, displaying rare determination at the crease and much of his old mastery with the ball.

Compound 23, 2- 1H-imidazol-1-yl -1- 4-{[3(trifluoromethoxy)benzyl]oxy}phenyl) ethanone, was the most interesting inhibitor of the series displaying a high potency at CYP11B1 (IC50 = 15 nM), increased selectivities over CYP11B2- 1H-imidazol-1-yl -1- 4-{[90) and CYP17 (5% inhibition at 2- 1H-imidazol-1-yl -1- 4-{[

Radioligand binding assay, performed on guinea pig brain membranes, identified 25b (1- 1,4-dioxaspiro[4.5]decan-2-ylmethyl -4-benzylpiperazine) as the most interesting compound of the series, displaying high affinity and selectivity for σ1- 1,4-dioxaspiro[4.5]decan-2-ylmethyl -4-benzylpiperazine

However, this process is highly relevant for lead optimization because it is not uncommon that a compound series displaying a promising SAR has other liabilities, e.g. toxic side effects.

Such SAR transfer series displaying similar target-specific SAR behavior are often sought after in medicinal chemistry as alternative compounds for optimization.

The series displayed low toxicity on five different cell lines.

The best compounds from the series displayed low nanomolar inhibitory activity and are selective versus PDE4.

The series displays her gentle humor, along with a wealth of sly social observations about 19th-century country life.

Both series displayed very good activity as well as selectivity towards the acetins within a short reaction time.

However, at similar density, the three polymers series displays a clear compliance drop that follows the increasing ESCR hierarchy.