Sentence examples for potency on the from inspiring English sources
The low in vitro effectiveness of the methylated inhibitors on the one hand and their high in vivo potency on the other hand is likely due to their high cellular permeability and the rapid cleavage of the methyl residue in planta, probably by a lipase (peak P1 in Figure 5).
Sessegnon missed a great chance to equalise when he raced on to Redmond's loose pass but dragged his shot wide when one on one with Ruddy and, as West Brom poured forward, Norwich's potency on the counter-attack grew.
The elongated trifluoroethoxy analogue 32 showed improved potency on the mouse orthologue.
Although the human and mouse receptor orthologues are closely related they are not identical and succinate shows a small increase in potency on the mouse receptor2.
Structure activity relationships within this series, leading to an increase of potency on the enzyme, is presented.
That does not look like the sort of message that will have any potency on the Arab street in the light of what is happening.
Our data show that CM and cocaine have very different potencies on the major cocaine targets, and therefore, equimolar systemic doses of CM do not produce equivalent inhibition of major cocaine targets.
The TEF system was developed based on relative potencies on the basis of intake, not tissue concentration.
Comparable enhancement of IGABA through α1β2 receptors as through the α1β2γ2S [3] and the similar potencies on the two receptor subtypes suggests that piperine interacts with a binding site located on α and/or β subunits.
The exploration led to development of potent drug-like, non-metabolite tool compounds with nanomolar potency on both the human and murine receptor orthologues and excellent physicochemical and in vitro stability properties.
Interestingly, and despite reduced agonist potency on CXCR4, the sustained binding of CXCL12γ to HS enabled it to promote in vivo intraperitoneal leukocyte accumulation and angiogenesis in matrigel plugs with much higher efficiency than CXCL12α.
