Sentence examples for is relatively potent from inspiring English sources

These studies resulted in the discovery of C646, a small molecule inhibitor of p300/CBP that is relatively potent, specific, and cell permeable.

The compound is relatively potent in inhibiting PV2 and PV3 replication, but has no activity against PV1, which limits its potential for PV.

It is relatively potent against p300 (IC50 of 750 nM) but not Pcaf (no detectable inhibition at 5 μM), and also inhibits acetylation in cells (ED50 of 5 μM by immunoblotting against acetyl-K9/K14 H3 in HepG2 cells).

In vitro studies indicated that most of these compounds are relatively potent inhibitors of each enzyme.

Third, this interaction should be achieved at low concentrations, meaning that the substance has to be relatively potent.

However, the best inhibitor in the cell culture model, compound 3624, was relatively potent in the second YopE secretion assays (60% at 10 µM).

Contact angles observed for the control proteins BSA and MBP (both at the relatively high concentration of 1 mg/mL) were very similar to those for buffer, suggesting that the effects observed for PLUNC were relatively potent and specific to that protein.

Budesonide, dexamethasone and prednisolone are known to be relatively potent, whilst betamethasone is known to be moderately potent.

These compounds are characterized as being relatively potent and selective toward a relatively narrow array of kinase targets.

Upon isolation the active compound was found to be in low abundance, indicating that it was relatively potent.

S1P was relatively potent, causing one-half maximal desensitization of GC-B at concentrations of 5 10 nM.