Sentence examples for increase its potency from inspiring English sources

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Supporters say that improvements upon the 1970s policy would increase its potency.

The drug was mixed with heroin to increase its potency, and resulted in more than 1,000 deaths, mostly of heroin users who were unaware that the drug contained fentanyl, or how potent it would be.

The next step, therefore, is for chemists to fiddle with the exact arrangement of a promising compound's atoms (subtracting one or two here, adding a few others there, in the way that Hoffmann did when he acetylated salicylic acid) in order to increase its potency.The "lead compound" which results from this tinkering is then subjected to further tests, this time generally in animals.

From these results, the preferential effect of 20d on non-phosphorylated VEGFR2 is dominated by its slow dissociation from the enzyme and this characteristically long residence time may increase its potency in vivo.

A series of 4EGI-1-derived thiazol-2-yl hydrazones have been designed and synthesized in order to delineate the structural latitude and improve its binding affinity to eIF4E, and increase its potency in inhibiting the eIF4E/eIF4G interaction.

Dexter: "Divorcing coaching and supervision from line management, whether internal or external, increases its potency.

A structure activity relationship study showed that a fluoro group on the phenyl ring greatly increased its potency and selectivity.

Here we report that N-methylation of 1a greatly increases its potency and results in excellent selectivity for SIRT2 over SIRT1 and SIRT3 isoforms.

An inhibitor of the complex of factor VIIa and tissue factor (fVIIa/TF), 2-substituted-4-amidinophenylpyruvic acid 1a, was structurally modified with the aim of increasing its potency and selectivity.

This indicates the importance of the LBD for the efficacy of enfuvirtide, as the octylation of enfuvirtide also increased its potency.