Sentence examples for inactive entry from inspiring English sources

However, this compound turned out to be biologically inactive (entry 1, Table 4).

N,N-dimethylalloxan (3 b) was found to be inactive (entry 3) despite possessing structural similarity to 3 a.

If the HO substituents in the hit compound 1a were substituted by fluorines the activity was slightly improved (IC50 = 75 μM, 1m, entry 13), whereas the corresponding Cl-analog 1n was inactive (entry 14) as also its structural isomer (entry 15).

Inactive compounds in CR assays were kept as inactive entries.

Although hydrazide 10 is a structurally very close analog to the active hydrazone 1b (Table 1) the hydrazone/hydrazide switch resulted in an inactive compound (entry 2, Table 4).

From the data of the first screening it also became apparent, that bulky substituents or multiple substitution leading to sterically demanding compounds resulted in inactive compounds (entries 9 12 and 20 26).

Compound C5 was furthermore evaluated, since demethylation of the quinoline methoxy group could reveal a stabilizing hydrogen-bond-donor functionality, but this was also found to be completely inactive (Table 2, entry 16).

Although members of the sample were identified as "inactive" at last entry into the Masterfile, 584 (37.0%) reported they were currently active in medicine at the time of our survey, and of these, 358 reported that they had not taken a leave from medicine of 6 months or more.

The RMSD (root mean square deviation) between α carbon positions in these two structures was 1.30 Å, and the α carbon RMSD for overlay of our inactive structure with PDB entry 3GT8 [ 20] was 1.42 Å.

In a hypothetical randomized controlled clinical trial with placebo (n = 100) and active (n = 100) groups, we assumed that each patient had 10 hypothetical latent lesions in their brain and that the lesions were in the inactive phase at the entry time.

Surprisingly, docking erlotinib into a crystal structure of the inactive EGFR-TKD (PDB entry 1XKK [ 13]), after removing lapatinib from the model, yielded a very similar Glide [ 32] score (−9.72 kcal/mol) to that seen for active EGFR-TKD (−9.34 kcal/mol).