Sentence examples for binding of the active from inspiring English sources

For estimating changes in TF activity, experimental assays may be employed based on the binding of the active form of the TF with a target reporter molecule.

As opposed to heparin, LMWLs significantly alter the binding of the active site fluorescent ligand p-aminobenzamidine.

We describe herein the development of a resin-immobilized, broad-spectrum synthetic MMP inhibitor for selective binding of the active forms of MMPs from different experimental samples.

To control release, it is necessary to rely on binding of the active agent to collagen, either by covalent or non-covalent bonds, or on sequestering in a secondary matrix.

Moreover, the binding energy of fucosterol and fucoxanthin was negative (−10.1 and −7.0 kcal/mol), indicating that hydrogen bonding may stabilize the open form of the enzyme and potentiate tight binding of the active site of BACE1, resulting in more effective BACE1 inhibition.

So the displacement binding of the active herbal components should be taken into consideration in the compatibility of TCMs, so as not to affect the efficacy.

A reaction of the pollutants with the components is also conceivable preventing binding on the active site of the enzyme.

It has been shown previously that Gly and Asp are inhibitors of AGA31,32 and thus capable of directly binding to the active site of AGA.

Energetics of cooperative ligand binding to the active sites of biosynthetic threonine deaminase from Escherichia coli.

The free energy of FRF substrate binding to the active site of human cathepsin L was equal to -7.5 to - 7.7 kcal/mol (Table  5).

Based on these, we postulated that the bioactive diterpenoid might exhibit anti-neuroinflammatory activities by binding to the active cavities of iNOS.