Sentence examples for binding activity of compound from inspiring English sources

This resulted in a sixfold decrease in binding activity of compound 1 b, 24 μ m (6 e, 275 μ m), a threefold decrease in binding activity of compound 7 g, 27 μ m (6 k, 68 μ m) and a twofold further decrease in binding activity of the already very weak blocker 7 a, 230 μ m (6 d, 481 μ m).

As shown in Figure 6A, the competitive binding activity of all compounds tested is dose-dependent.

Minimal differences in the affinities were observed compared to data obtained using DDM detergent suggesting a very limited influence of the different detergents on binding activity of the compounds.

Thus, we evaluated the binding activities of silagaba compounds to the gabapentin-binding sites, presumably α2-δ subunit proteins, in rat brain cortex by means of [H]gabapentin-binding assay.

Compounds were tested for their ability to displace EtBr from DNA as an indication of the DNA-binding activity of each compound.

Here fluorescence binding assay was used to determine the binding activity of AfunOBP1 and AfunOBP3 to the EAG-active compounds.

Among these novel inhibitors, compound SC7 was found to inhibit the DNA binding activity of the EBNA1 protein in FP assays with an IC50 value of 23 µM.

Binding activity of dust samples.

Encouragingly, a dose-dependent reduction in the DNA-binding activity of STAT3 was observed in the presence of compound 1.

The chemometric statistical analysis infers differences of binding activity for sets of compounds against TIR1 and AFB5.

A dose-response experiment was performed to determine the potency of compound 1 at inhibiting the DNA-binding activity of STAT3.