Sentence examples for being a partial agonist from inspiring English sources

These agonist/antagonist results are consistent with TCS being a partial agonist of the AhR.

Thus, telmisartan being a partial agonist of PPAR- γ justifies the significant decreased in serum glucose levels.

Thus, telmisartan being a partial agonist of PPAR- γ justifies the significant increase in food intake which accounts for the increased body weight.

This suggested that while GH RFP GPI differed from GH GPI and GH LL GPI by being a partial agonist, it shared with the other GPI constructs the ability to block the action of exogenously administered GH.

Thus, telmisartan being a partial agonist of PPAR- γ justifies the significant decreased in serum insulin levels, suggesting that addition of telmisartan to cisplatin treatment may prevent insulin resistance mediated protein degradation and skeletal muscle wasting.

Tamoxifen acts by blocking the ER but under certain circumstances can change to being a partial agonist via the ER and this may limit its preventive utility since in some women at increased risk it appears to increase mammographic density [ 127].

Just as bupe is a "partial agonist" of opiate receptors, Chantix partially binds to nicotinic receptors, reducing cravings while simultaneously making smoking less pleasurable.

Varenicline is a partial agonist at alpha4beta2 and a full agonist at alpha7 neuronal nicotinic receptors.

Because it is a partial agonist, it has a ceiling effect.

Cytisine is a partial agonist at α4β2* and α6β2* nAChRs and a full agonist at α3β4* and α7 nAChRs (Salminen et al, 2004; Grady et al, 2010).

This medication (Subutex) is a partial agonist for opioid receptors, which means it is less efficient than a medication like methadone.