Sentence examples for antagonistic activity from inspiring English sources
It has antagonistic activity at the glucocorticoid receptor especially with reduced receptors number [ 17].
The antagonistic activity of LBD, but not NRR, antibodies is strongly dependent on the activating ligand.
In contrast, six analogues presented antagonistic activity.
Representative compound 3a exhibits PPARδ-preferential antagonistic activity.
Despite this similarity, bosentan sterically prevents the inward movement of transmembrane helix 6 (TM6), and thus exerts its antagonistic activity.
The triamine derivative with a guanidine moiety showed more potent antagonistic activity than memantine.
Several tricyclic compounds showed potent antagonistic activity in rat AVP receptors V1a and V2.
The aminoadamantane derivatives exhibited similar NMDA antagonistic activity to amantadine 1.
Moreover, strain AR6 exhibited strong antagonistic activity against phytopathogen Aspergillus niger.
The (2S,3R) configuration of the pyrrolidine ring was favorable for the AR antagonistic activity.
Further, its putative metabolite (12a) exhibited potent ERα-antagonistic activity (IC50 = 29.7 nM).
