Sentence examples for antagonist without from inspiring English sources
Consequently, 4-[ 5-chlorothiophen-2-yl)methoxy]-1-(2-cyclopropyl-1-methyl-1H-benzimidazol-6-yl)pyridin-2(1H)-one (6s) was identified as a potent MCHR1 antagonist without the risk of CYP3A4-[ 5-chlorothiophen-2-ylpromising safety profile including low CYP3A4-[ 5-chlorothiophen-2-ylsignificant antiobesity effects in diet-induced obese F34-[ 5-chlorothiophen-2-yl
Treatment involved the sole use of tamoxifen, an oestrogen-receptor antagonist, without surgery, radiotherapy or chemotherapy.
Granisetron is a selective of 5HT3 receptor antagonist without relevant affinity to other serotonin receptors.
This finding also increase the evidence of the atypical properties of amisulpride, despite its action as D2/D3 antagonist without affinity with other neurotransmitter systems.
One of the older, but still frequently prescribed topical drugs is timolol, which is a non-selective beta-adrenoceptor antagonist without intrinsic sympathicomimetic activity.
In this study, a new dosage format of cisplatin is introduced combining the advantages described above (high dose, embolization, high response, low toxicity, use of antagonist) without the drawbacks.
We have been developing partial CXCR4 antagonists without such property.
Compounds 24b and 25b are strong RARα,β-selective antagonists without agonist or antagonist activities for RARγ.
No significant eruption occurred in unopposed mandibular second molars bonded with fixed sectional retainers compared to molars partially occluded with the antagonists without fixed retention.
Various 4- anilino pyrrole-2-carboxamides were designed and synthesized as novel androgen receptor (AR) antagonists without steroidal or anilide structure, based on our strategy for developing full antagonists of nuclear receptors.
This method could be used as an helpful general procedure for the design of novel A3 adenosine receptor antagonists without the difficulty of separating the N8-substituted pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines from the corresponding N7-isomers.
